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NCT03195699 · ClinicalTrials.gov registry record · Phase 1

Oral STAT3 Inhibitor, TTI-101, in Patients with Advanced Cancers

A Phase 1 study of Breast Cancer and Non-Small Cell Lung Cancer, sponsored by Tvardi Therapeutics, Incorporated.

Completed
Registry status
Phase 1
Development phase
64
Enrollment target
2
Study locations

NCT03195699: Completed Phase 1 study of Breast Cancer and Non-Small Cell Lung Cancer, sponsored by Tvardi Therapeutics, Incorporated.

NCT03195699 is a Phase 1 study of Breast Cancer and Non-Small Cell Lung Cancer that has completed, run by Tvardi Therapeutics, Incorporated. The registered enrollment target is 64 participants, below the 2,803-participant average among 1,224 other Breast Cancer trials with a reported enrollment target (98% lower). The trial reports 2 study locations across 1 state. According to ClinicalTrials.gov, the official US trial registry.

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The verdict

NCT03195699, a Phase 1 study of Breast Cancer and Non-Small Cell Lung Cancer, has completed, sponsored by Tvardi Therapeutics, Incorporated.

COMPLETED
Registry status
Phase 1
Development phase
64 participants
Enrollment target
2
Study locations

Study Summary

Many patients have cancers that have increased activity of a protein called STAT3 that contributes critically to the development and growth of their cancer. Despite our knowledge of STAT3's importance to cancer, scientists and doctors have not developed a drug that targets it and that patients can take to treat their cancer more effectively than treatments that are now available. Tvardi Therapeutics, Incorporated has developed a compound, TTI-101, which can be given by mouth and acts as a direct inhibitor of STAT3. Administration of TTI-101 to mice demonstrated that it blocked growth of cancers of the breast, head and neck, lung, and liver and it was safe when administered at high doses to mice, rats, and dogs. In this application, Tvardi is proposing to further develop TTI-101 for treatment of solid tumors for which the prognosis is dismal. The investigators will determine how safe it is when administered to patients with cancer, determine whether an adequate dose can be administered to patients with cancer that will block STAT3 in their cancer, and determine whether treatment with TTI-101 leads to reduced growth of their cancer.

Primary Outcome

To determine the maximum tolerated dose (MTD), dose-limiting toxicities, and tolerability of TTI-101 administered orally to patients with advanced breast cancer and other solid tumors. Dose-limiting toxicity is defined as a Grade 3 or above adverse event (using CTCAE v5.0) within the first treatment cycle (28-days).

Interventions

  • DRUG TTI-101

Study Locations (2)

Texas

  • The University of Texas MD Anderson Cancer Center - Houston
  • Mays Cancer Center at University of Texas Health Science Center SA - San Antonio

Trial Details

FieldValue
Enrollment Target 64 participants
Start Date 2017-11-15
Est. Completion 2024-06-24
Phase Phase 1

What the finished NCT03195699 record still lists

NCT03195699 is an interventional study that assigns participants to a tested intervention. The registry caps enrollment at 64 participants, a relatively small participant target, below the 2,803-participant average among 1,224 other Breast Cancer trials with a reported enrollment target (98% lower).

The record links to 8 conditions, with Breast Cancer appearing as the primary indexed condition, and to 1 intervention - of which TTI-101 is the first listed.

NCT03195699 reports a single indexed study location in Texas.

Frequently Asked Questions

What is clinical trial NCT03195699 about?

NCT03195699 is a clinical study titled "Oral STAT3 Inhibitor, TTI-101, in Patients with Advanced Cancers". Many patients have cancers that have increased activity of a protein called STAT3 that contributes critically to the development and growth of their cancer. Despite our knowledge of STAT3's importance to cancer, scientists and doctors have not developed a drug that targets it and that patients can t...

What is the current status of trial NCT03195699?

This trial is currently completed. It is a Phase 1 study. The enrollment target is 64 participants. The study started on 2017-11-15. Estimated completion is 2024-06-24.

What conditions does trial NCT03195699 study?

This clinical trial studies the following conditions: Breast Cancer, Non-Small Cell Lung Cancer, Colorectal Cancer, Melanoma, Head and Neck Squamous Cell Carcinoma.

What interventions are being tested in trial NCT03195699?

The interventions under investigation include: TTI-101 (DRUG).

Who is sponsoring clinical trial NCT03195699?

This trial is sponsored by Tvardi Therapeutics, Incorporated, which has 4 total clinical trials registered on ClinicalTrials.gov.

Where is trial NCT03195699 being conducted?

This trial has 2 study locations across Texas. Contact the study sites directly through ClinicalTrials.gov for enrollment availability.

Similar trials for Breast Cancer

Matched on the same primary condition, ranked to surface studies in the same phase first, then by recruiting status, no relevance scoring or editorial curation.

Where NCT03195699's enrollment target sits among peer trials

64 725th of 1224 higher than 499 of 1,224 other Breast Cancer trials

participants (enrollment target), bucketed by value

Each bar is a band; taller bars hold more other Breast Cancer trials. The dashed line + filled bar mark this entry. Hover or tap any bar for its full count and share, and where it sits relative to this entry.

Source ClinicalTrials.gov registry export · 2026-08-08

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Source: ClinicalTrials.gov NCT03195699, the US trial registry maintained by the National Library of Medicine. NCT03195699 (small enrollment · single site footprint · completed) retrieved and formatted by PlainTrial, see methodology.