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NCT01981499 · ClinicalTrials.gov registry record · Phase 1

A Study of the Safety, Tolerability, Pharmacokinetics, And Effects On Histamine-Induced Wheal Of PF-05180999 In Healthy Adults

A Phase 1 study, sponsored by Pfizer.

Terminated
Registry status
Phase 1
Development phase
31
Enrollment target

NCT01981499: Clinical Trial Phase 1 study, sponsored by Pfizer.

NCT01981499 is a Phase 1 study that was terminated before completion, run by Pfizer. The registered enrollment target is 31 participants, below the 60-participant average among 29,502 other Phase 1 trials with a reported enrollment target (48% lower). According to ClinicalTrials.gov, the official US trial registry.

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The verdict

NCT01981499, a Phase 1 study, was terminated before completion, sponsored by Pfizer.

TERMINATED
Registry status
Phase 1
Development phase
31 participants
Enrollment target

Study Summary

PF-05180999 is a phosphodiesterase-2 inhibitor that is hypothesized to be able to reduce vascular permeability. The purpose of this study is to evaluate the safety, tolerability, pharmacokinetics, and effects on histamine-induced wheal of single doses of PF-05180999 in healthy adult subjects. Histamine-induced wheals are biomarkers of vascular permeability.

Primary Outcome

Maximum observed plasma concentration

Interventions

  • DRUG Placebo
  • DRUG PF-05180999
  • DRUG 120 mg MR PF-05180999
  • DRUG 360 mg MR PF-05180999
  • DRUG 10 mg cetirizine

Trial Details

FieldValue
Enrollment Target 31 participants
Start Date 2014-01
Est. Completion 2014-04
Phase Phase 1
Pfizer

1,845 total trials

Why NCT01981499 stopped before completion

NCT01981499 is an interventional study that assigns participants to a tested intervention. The registry caps enrollment at 31 participants, a relatively small participant target, below the 60-participant average among 29,502 other Phase 1 trials with a reported enrollment target (48% lower).

The record links to 0 conditions, and to 5 interventions - of which Placebo is the first listed.

NCT01981499 does not publish any study locations in the registry export this page uses.

Frequently Asked Questions

What is clinical trial NCT01981499 about?

NCT01981499 is a clinical study titled "A Study of the Safety, Tolerability, Pharmacokinetics, And Effects On Histamine-Induced Wheal Of PF-05180999 In Healthy Adults". PF-05180999 is a phosphodiesterase-2 inhibitor that is hypothesized to be able to reduce vascular permeability. The purpose of this study is to evaluate the safety, tolerability, pharmacokinetics, and effects on histamine-induced wheal of single doses of PF-05180999 in healthy adult subjects. Histam...

What is the current status of trial NCT01981499?

This trial is currently terminated. It is a Phase 1 study. The enrollment target is 31 participants. The study started on 2014-01. Estimated completion is 2014-04.

What interventions are being tested in trial NCT01981499?

The interventions under investigation include: Placebo (DRUG), PF-05180999 (DRUG), 120 mg MR PF-05180999 (DRUG), 360 mg MR PF-05180999 (DRUG), 10 mg cetirizine (DRUG).

Who is sponsoring clinical trial NCT01981499?

This trial is sponsored by Pfizer, which has 1,845 total clinical trials registered on ClinicalTrials.gov.

How this trial's enrollment target compares

Where NCT01981499's enrollment target sits among peer trials

31 1322nd of 2000 higher than 669 of 2,000 other Phase 1 trials

participants (enrollment target), bucketed by value

Each bar is a band; taller bars hold more other Phase 1 trials. The dashed line + filled bar mark this entry. Hover or tap any bar for its full count and share, and where it sits relative to this entry.

Source ClinicalTrials.gov registry export · 2026-08-08

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Source: ClinicalTrials.gov NCT01981499, the US trial registry maintained by the National Library of Medicine. NCT01981499 (small enrollment · none site footprint · terminated) retrieved and formatted by PlainTrial, see methodology.