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NCT02289482 · ClinicalTrials.gov registry record · Phase 1

A Single Dose Pharmacokinetic (PK) and Safety Study of GSK2838232 With and Without Ritonavir (RTV) Conducted in Healthy Subjects

A Phase 1 study, sponsored by GlaxoSmithKline.

Terminated
Registry status
Phase 1
Development phase
20
Enrollment target

NCT02289482: Clinical Trial Phase 1 study, sponsored by GlaxoSmithKline.

NCT02289482 is a Phase 1 study that was terminated before completion, run by GlaxoSmithKline. The registered enrollment target is 20 participants, below the 60-participant average among 29,502 other Phase 1 trials with a reported enrollment target (67% lower). According to ClinicalTrials.gov, the official US trial registry.

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The verdict

NCT02289482, a Phase 1 study, was terminated before completion, sponsored by GlaxoSmithKline.

TERMINATED
Registry status
Phase 1
Development phase
20 participants
Enrollment target

Study Summary

This study investigates the safety, tolerability and PKs of GSK2838232 with and without Ritonavir, and to evaluate different formulations of GSK2838232 in healthy subjects. This study will evaluate higher single and RTV boosted doses to support continued clinical development of GSK2838232 at clinically relevant doses, and subsequently in those infected with HIV in a dose ranging phase 2 study. The study is conducted in 2 parts: Part A and Part B, study Part A and Part B may be conducted in parallel. Approximately 20 healthy subjects will be enrolled into the study, 8 in Part A and 12 in Part B. Part A is a double-blind, randomized, placebo-controlled, 4-period, single dose escalation design. Subjects will be randomized 3:1 to receive GSK2838232 or placebo. Subjects randomized to placebo will receive placebo in all four periods. Following completion of Period 2 PK assessments at 96hr post-dose, subjects will begin daily dosing of RTV 100mg for a total of 26 days. Part B is a randomized, open-label, unbalanced, 3-period, cross-over design; subjects will be randomized 1:1 to each sequence. The relative bioavailability of single 100mg doses of powder in a bottle (PIB) active pharmaceutical ingredient (API) of GSK2838232 versus PIB spray-dried dispersion (SDD) will be assessed. A single dose of GSK2838232 will co-administered on the 10th day of RTV dosing; RTV dosing will continue for an additional 4 days (total of 14 days). Subjects will have a screening visit within 30 days prior to first dose and a follow-up visit 7-14 days after the last dose.

Primary Outcome

Safety was assessed by monitoring AE and serious AEs (SAE). AEs and SAEs will be collected from the start of Study Treatment until the follow-up contact

Interventions

  • DRUG Placebo
  • DRUG Ritonavir
  • DRUG GSK2838232 PIB (SDD)
  • DRUG GSK2838232 PIB (API)

Trial Details

FieldValue
Enrollment Target 20 participants
Start Date 2014-11-17
Est. Completion 2015-03-10
Phase Phase 1
GlaxoSmithKline

1,345 total trials

Why NCT02289482 stopped before completion

NCT02289482 is an interventional study that assigns participants to a tested intervention. The registry caps enrollment at 20 participants, a relatively small participant target, below the 60-participant average among 29,502 other Phase 1 trials with a reported enrollment target (67% lower).

The record links to 0 conditions, and to 4 interventions - of which Placebo is the first listed.

NCT02289482 does not publish any study locations in the registry export this page uses.

Frequently Asked Questions

What is clinical trial NCT02289482 about?

NCT02289482 is a clinical study titled "A Single Dose Pharmacokinetic (PK) and Safety Study of GSK2838232 With and Without Ritonavir (RTV) Conducted in Healthy Subjects". This study investigates the safety, tolerability and PKs of GSK2838232 with and without Ritonavir, and to evaluate different formulations of GSK2838232 in healthy subjects. This study will evaluate higher single and RTV boosted doses to support continued clinical development of GSK2838232 at clinica...

What is the current status of trial NCT02289482?

This trial is currently terminated. It is a Phase 1 study. The enrollment target is 20 participants. The study started on 2014-11-17. Estimated completion is 2015-03-10.

What interventions are being tested in trial NCT02289482?

The interventions under investigation include: Placebo (DRUG), Ritonavir (DRUG), GSK2838232 PIB (SDD) (DRUG), GSK2838232 PIB (API) (DRUG).

Who is sponsoring clinical trial NCT02289482?

This trial is sponsored by GlaxoSmithKline, which has 1,345 total clinical trials registered on ClinicalTrials.gov.

How this trial's enrollment target compares

Where NCT02289482's enrollment target sits among peer trials

20 1629th of 2000 higher than 285 of 2,000 other Phase 1 trials

participants (enrollment target), bucketed by value

Each bar is a band; taller bars hold more other Phase 1 trials. The dashed line + filled bar mark this entry. Hover or tap any bar for its full count and share, and where it sits relative to this entry.

Source ClinicalTrials.gov registry export · 2026-08-08

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Source: ClinicalTrials.gov NCT02289482, the US trial registry maintained by the National Library of Medicine. NCT02289482 (small enrollment · none site footprint · terminated) retrieved and formatted by PlainTrial, see methodology.